KPH2f 是一种安全、口服有效的URAT1/GLUT9双抑制剂，对 URAT1 和 GLUT9 的 IC50分别为 0.24 μM 和 9.37 μM。KPH2f 对 OAT1 和 ABCG2 几乎没有影响 (IC50分别为 32.14 和 26.74 μM)。

KPH2f is a safe, orally active, and effective dual URAT1/GLUT9 inhibitor with IC 50 s of 0.24 μM and 9.37 μM for URAT1 and GLUT9, respectively. KPH2f shows little effects on OAT1 and ABCG2 (IC 50 =32.14 and 26.74 μM) [1].

C24H16N3NaO2S

433.46

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years