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Azimilide Dihydrochloride
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Azimilide Dihydrochloride图片
CAS NO:149888-94-8
包装与价格:
包装价格(元)
5 mg电议
10 mg电议
50 mg电议
100 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
盐酸阿齐利特
NE-10064 Dihydrochloride
产品介绍
Azimilide dihydrochloride 是 I(Ks) 和 I(Kr) 抑制剂,具有抗心律失常活性。

产品描述

Azimilide Dihydrochloride, a novel class III antiarrhythmic agent, blocks both the slowly activating (IKs) and rapidly activating (IKr) components of the delayed rectifier potassium current

体内活性

Azimilide has shown excellent efficacy (>85%) in suppressing supraventricular arrhythmias in a variety of dog models.?It also suppressed complex ventricular arrhythmias in infarcted dogs and, in a sudden death cardiac model, decreased mortality[1].

Cas No.

149888-94-8

分子式

C23H30Cl3N5O3

分子量

530.88

别名

盐酸阿齐利特;NE-10064 Dihydrochloride

储存和溶解度

DMSO:8.46 mg/mL (15.94 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years