TC-E 5003 是选择性PRMT1抑制剂,其IC50值为1.5 μM。它在 TLR4 信号传导中具有抗炎特性。
产品描述
TC-E 5003 is a selective inhibitor of PRMT1 with IC50 of 1.5 μM.
体外活性
The GI50 values for TC-E 5003 were 1.97 μM on MCF7a cells and 4.49 μM on LNCaP cells.
Cas No.
17328-16-4
分子式
C16H14Cl2N2O4S
分子量
401.26
别名
NSC 30176;TC-E 5003
储存和溶解度
DMSO:45mg/ml(112.15mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years