VU 0255035 是高度选择性、竞争性和血脑屏障通透性的毒蕈碱 M1 受体拮抗剂,IC50为 130 nM,可减少毛果芸香碱诱导的小鼠癫痫发作。
产品描述
VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM. It reduces pilocarpine-induced seizures in mice. It is used to examine the role of the M1 receptor in diverse situations.
Cas No.
1135243-19-4
分子式
C18H20N6O3S2
分子量
432.52
别名
VU 0255035
储存和溶解度
DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years