Nitrocaramiphen hydrochloride 是一种选择性 M1 毒蕈碱拮抗剂,可抑制与大脑中 sigma 位点的结合。
产品描述
Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.
体外活性
Nitrocaramiphen hydrochloride binds with high affinity for M1 sites (Ki = 5.5 nM) and with a 71-fold selectivity over M2, and a 10-fold selectivity for the M1 over the M3 subtype[1].?
Cas No.
98636-73-8
分子式
C18H27ClN2O4
分子量
370.87
别名
Nitrocaramiphen hydrochloride
储存和溶解度
H2O:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years