Pimethixene 是抗组胺和抗血清素剂,用作抗偏头疼剂。它是高效多靶点拮抗剂。
产品描述
Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
Cas No.
314-03-4
分子式
C19H19NS
分子量
293.43
别名
匹美噻吨;Calmixen;Pimetixene;Pimethixene
储存和溶解度
DMSO:18.33 mg/ml (62.48 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years