Brimonidine 是一种完全的α2肾上腺素受体激动剂。

Brimonidine is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertension

[3H]Brimonidine is a full agonist at alpha 2-adrenergic receptors labeling at least 2 specific binding sites in the human brain that both have the characteristics of an alpha 2-adrenergic binding site. GTP decreases agonist binding at both of these sites, but with different potencies at each site [1].

59803-98-4

C11H10BrN5

292.14

溴莫尼定;Bromoxidine;AGN 190342;AGN-190342;AGN190342;Brimonidine

DMSO:26 mg/mL (89.0 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years