Alpha-Methyldopa Sesquihydrate 是一种前药,在中枢神经系统中被代谢成 α-Methylepinephrine。它是一种 α-肾上腺素能激动剂,对α2-Adrenergic Receptors有选择性。
产品描述
Alpha-Methyldopa Sesquihydrate is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, norepinephrine, and epinephrine, and exhibits NO-dependent sedative activity.
Cas No.
41372-08-1
分子式
C20H32N2O11
分子量
476.479
别名
Alpha-Methyldopa Sesquihydrate;Methyldopa Sesquihydrate;MK-351 hydrate;L-甲基多巴;L-(-)-α-Methyldopa hydrate;Methyldopa hydrate
储存和溶解度
DMSO:33.33 mg/mL (139.90 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years