Relamorelin, formerly known as BIM28131 and RM131, is a centrally penetrant, selective agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) potentially useful for the treatment of diabetic gastroparesis, chronic idiopathic constipation, and anorexia nervosa. It is a pentapeptide and analogue of ghrelin with improved potency and pharmacokinetics. In humans, relamorelin produces increases in plasma growth hormone, prolactin, and cortisol levels, and, like other GHSR agonists, increases appetite.

纯度：≥98%

CAS：661472-41-9