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CAY10499
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CAY10499图片
包装与价格:
包装价格(元)
5 mg电议
10 mg电议
25 mg电议

产品介绍

产品描述

CAY10499 is a potent inhibitor of monoglyceride lipase (MGL) and human hormone-sensitive lipase. CAY10499 inhibited MGL-mediated 4-NPA hydrolysis with the IC 50 value of 0.5 ± 0.03 μM. CAY10499 fully inhibited [3H]-AEA hydrolysis by human recombinant FAAH with an IC50 of 76 nM. CAY10499 displaced only 25% and 20% of [3H]-CP-55940-specific binding to the CB1 and CB2 receptors, respectively [1]. CAY10499 potently inhibited the activity of human hormone-sensitive lipase with an IC50 of 90 nM for the recombinant human hormone-sensitive lipase enzyme [1][2].

Cas No.

T22637

分子式

C18H17N3O5

分子量

355.3

别名

CAY10499

储存和溶解度

DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years