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BMT-124110
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
BMT-124110图片
CAS NO:1679371-59-5
包装:5 mg
市场价:7000元

产品介绍

产品描述

BMT-124110 is an effectivet, selective AAK1 inhibitor (IC50: 0.9 nM) with antinociceptive activity. BMT-090605 inhibits BMP-2-inducible protein kinase (BIKE; IC50: 17 nM) and Cyclin G-associated kinase (GAK; IC50: 99 nM).

体外活性

BMT-124110 shows a cellular IC50 of 3.2 nM for AAK1.

体内活性

BMT-124110 is added directly onto the spinal covered by microiontophoresis, leading to a reduction in windup-induced activity in 10 of 14 animals.

Cas No.

1679371-59-5

分子式

C21H27N3O3

分子量

369.46

别名

BMT-124110

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years