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APC-6860
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CAS NO:154628-42-9
包装与价格:
包装价格(元)
5 mg电议
100 mg电议
500 mg电议

产品介绍

产品描述

APC-6860 is a trypsin-like serine proteases inhibitor with k i values of 0.21, 0.44, 1.5, 16.8, 20, 30 μM for uPA, trypsin, tryptase, tPA, thrombin and factor Xa, respectively. APC-6860 has a selectivity ratio for tPA versus uPA of 80. APC-6860 has k i values of 0.1, 0.082 μM for human and murine urokinases, respectively. APC-6860 can be used for the research of cancer.

体外活性

APC-6860 (compounds 2) inhibits urokinases in MiaPaCa-2 and Lewis Lung Carcinoma cells with IC 50 s of 1.4 and 3.1 μM, respectively[2].

Cas No.

154628-42-9

分子式

C9H7IN2S

分子量

302.13

别名

APC-6860

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years