Vildagliptin carboxylic acid metabolite is the major metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor vildagliptin in humans. Vildagliptin carboxylic acid metabolite has an IC50 value of 477 μM for DPP-4 in human Caco-2 cells. It is formed from hydrolysis of the cyano group on vildagliptin.

565453-41-0

C19H27F3N2O6

436.42

Vildagliptin carboxylic acid metabolite (trifluoroacetate salt)

DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years