Gü1303 是一种有效的、可逆的、慢结合的组织蛋白酶 K (CAThepsin K (CATK)) 抑制剂，对 成熟 CATK (mCATK) 的Ki值为 0.91 nM。Gü1303 抑制组织蛋白酶 K 酶原的自催化激活。

Gü1303 is a potent, reversible, slow-binding cathepsin K (CatK) inhibitor with a K i of 0.91 nM for mature CatK (mCatK). Gü1303 suppresses the autocatalytic activation of the cathepsin K zymogen [1].

1043922-53-7

C20H22N4O3

366.41

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years