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SSTR5 antagonist 2
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
SSTR5 antagonist 2图片
CAS NO:1254730-81-8
包装:5 mg
市场价:7000元

产品介绍

产品描述

SSTR5 antagonist 2 is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5),with potential to treat type 2 diabetes mellitus (T2DM).

体内活性

Both total and active circulating incretin hormone GLP1 levels in mice at a dose of 10 mg/kg increased by SSTR5 antagonist 2 (10 mg/kg, orally) . SSTR5 antagonist 2 increases pancreatic insulin secretion as well as total and active GLP1 release, and demonstrates synergistic effects in combination with DPP4 inhibitors.

Cas No.

1254730-81-8

分子式

C32H35FN2O5

分子量

546.63

别名

SSTR5 antagonist 2

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years