产品描述
Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM). Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. Recuces tumor expansion and lengthens survival time in a mouse xenograft model of glioblastoma.
Cas No.
1313027-43-8
分子式
C70H121N29O15S4
分子量
1737.15
别名
MM 54
储存和溶解度
H2O:2 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years