产品描述
Highly potent and selective NOP receptor agonist (EC50 = 1 nM). Displays >875-fold selectivity over opioid receptors (IC50 values are 0.32, 280, >10000 and 1500 for NOP, μ, δ and κ receptors respectively). Longer lasting and 30-fold more potent than nociceptin in vivo; pronociceptive and inhibits locomotor activity.
Cas No.
236098-40-1
分子式
C82H137N31O22
分子量
1909.18
别名
[Arg14,Lys15]Nociceptin
储存和溶解度
H2O:1 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years