PKC-IN-1 is a novel, potent, ATP-competitive and reversible inhibitor of conventional PKC enzymes (Kis = 5.3 and 10.4 nM for human PKCβ and PKCα, and IC50s = 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM for PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε, respectively).

纯度：≥98%

CAS：1046787-18-1