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Taltirelin acetate(TA0910 Ceredist)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Taltirelin acetate(TA0910 Ceredist)图片
CAS NO:1549593-23-8
规格:≥98%
包装与价格:
包装价格(元)
25mg电议
50mg电议
100mg电议
250mg电议
500mg电议

产品介绍

Taltirelin acetate (TA-0910; tradename Ceredist) is a thyrotropin-releasing hormone (TRH) analog and a TRH mimic that acts as a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release). Taltirelin alleviates mechanical allodynia through activation of descending monoaminergic neurons in persistent inflammatory pain. Compare to TRH, it has a much longer half-life and duration of effects, and little development of tolerance following prolonged dosing. It has nootropic, neuroprotective and analgesic effects

纯度:≥98%

CAS:1549593-23-8