Azidothiorphan is a photoaffinity ligand for the active site of the neutral endopeptidase 24.11. After ultraviolet irradiation the inhibitor binds irreversibly to the enzyme, and photolabeling occurs at the active site. The competitive inhibitor thiorphan protects the endopeptidase from inactivation. References: Beaumont A, Hernandez JF, Chaillet P, Crine P, Roques BP. irreversible (covalent) photolabeling of active site of neutral endopeptidase-24.11 'enkephalinase' by azidothiorphan and [14C]-azidothiorphan. Mol Pharmacol. 1987 Nov;32(5):594-9. PubMed PMID: 3479679.

纯度：≥98%

CAS：83960-29-6