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NS-304(Selexipag)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
NS-304(Selexipag)图片
CAS NO:475086-01-2
包装与价格:
包装价格(元)
10mg电议
25mg电议
50mg电议

产品名称
Selexipag, ACT-293987
产品介绍

生物活性

NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂(人和大鼠IP受体的Ki值为260和2100 nM,EP1-4,DP,FP和TP受体的Ki值为> 10μM)。

化学数据

目录号A13880
作用机制Agonist (激动剂)
M. Wt496.6
FormulaC26H32N4O4S
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.475086-01-2
SynonymsSelexipag, ACT-293987
SMILESCC(C)N(CCCCOCC(=O)NS(=O)(=O)C)C1=CN=C(C(=N1)C2=CC=CC=C2)C3=CC=CC=C3

溶解度

In vitroDMSO84 mg/mL (169.14 mM)
WaterInsoluble
Ethanol42 mg/mL (84.57 mM)
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM20.14 mL100.68 mL201.37 mL
0.5 mM4.03 mL20.14 mL40.27 mL
1 mM2.01 mL10.07 mL20.14 mL
5 mM0.4 mL2.01 mL4.03 mL

*The above data is based on the productmolecular weight 496.6. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.