MK-6240是一种针对神经纤维缠结(NFTs)的正电子发射断层显像(PET)示踪剂,对NFT的结合具有较高的特异性和选择性。
CAS:1841078-87-2
分子式:C16H11FN4
分子量:278.28
纯度:98%
存储:Store at -20°C
Background:
MK-6240 is a positron emission tomography (PET) tracer for neurofibrillary tangles (NFTs), exhibiting high specificity and selectivity for binding to NFTs.
[1]. Walji AM, et al. Discovery of 6-(Fluoro-(18)F)-3- (1H-pyrrolo [2,3-c]pyridin-1-yl) isoquinolin-5-amine ([(18)F]-MK-6240): A Positron Emission Tomography (PET) Imaging Agent for Quantification of Neurofibrillary Tangles (NFTs). J Med Chem. 2016 May 26;59(10):4778-89.