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Clemastine Fumarate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Clemastine Fumarate图片
CAS NO:14976-57-9
包装与价格:
包装价格(元)
100mg电议
250mg电议
10mM * 1mL in DMSO电议

产品名称
Meclastin
产品介绍

生物活性

Clemastine fumarate是一种选择性的组胺H1拮抗剂。它与组胺H1受体结合,从而阻断了内源性组胺的作用,从而暂时缓解了由组胺引起的阴性症状。

靶点信息

Histamine H1 receptor
3 nM

化学数据

目录号A10226
M. Wt459.96
FormulaC21H26ClNO.C4H4O4
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.14976-57-9
Synonymsmeclastin
SMILESC[C@@](C1=CC=CC=C1)(C2=CC=C(C=C2)Cl)OCC[C@H]3CCCN3C.C(=C/C(=O)O)\C(=O)O

溶解度

In vitroDMSOWarmed: 31 mg/mL (67.39 mM)
WaterInsoluble
EthanolInsoluble
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM21.74 mL108.71 mL217.41 mL
0.5 mM4.35 mL21.74 mL43.48 mL
1 mM2.17 mL10.87 mL21.74 mL
5 mM0.43 mL2.17 mL4.35 mL

*The above data is based on the productmolecular weight 459.96. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.