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Risperidone(Risperdal)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Risperidone(Risperdal)图片
CAS NO:106266-06-2
包装与价格:
包装价格(元)
10mg电议
50mg电议
100mg电议
200mg电议

产品名称
R 64 766, Risperdal
产品介绍

生物活性

Risperidone (Risperdal)是一种非典型的抗精神病药,用于治疗精神分裂症(包括青少年精神分裂症),精神分裂症,躁郁症的躁狂和躁狂状态,以及自闭症儿童的烦躁不安。

Targets

TargetValue
5-HT2Aki: 0.17nM
α2c-adrenergicreceptorki: 1.3nM
D2receptorki: 3.57nM
D3receptorki: 3.6nM
D2LReceptorki: 4.16nM
D4receptorki: 4.66nM
D2SReceptorki: 4.73nM
α1A-adrenergicreceptorki: 5nM
5-HT7ki: 6.6nM
α1B-adrenergicreceptorki: 9nM
5-HT2Cki: 12nM
5-HT1Bki: 14.9nM
α2a-adrenergicreceptorki: 16.5nM
H1receptorki: 20.1nM
5-HT2Bki: 61.9nM
5-HT1Dki: 84.6nM
α2b-adrenergicreceptorki: 108nM
H2receptorki: 120nM
5-HT5Aki: 206nM
5-HT5Aki: 206nM
D1receptorki: 244nM
D5receptorki: 290nM
5-HT1Aki: 423nM
5-HT6ki: 2060nM

化学数据

目录号A10797
M. Wt410.5
FormulaC23H27FN4O2
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.106266-06-2
SynonymsR 64 766, Risperdal
SMILESCC1=C(C(=O)N2CCCCC2=N1)CCN3CCC(CC3)C4=NOC5=C4C=CC(=C5)F

溶解度

In vitroDMSOWarmed: 4 mg/mL (9.74 mM)
WaterInsoluble
Ethanol4 mg/mL (9.74 mM)
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM24.36 mL121.8 mL243.61 mL
0.5 mM4.87 mL24.36 mL48.72 mL
1 mM2.44 mL12.18 mL24.36 mL
5 mM0.49 mL2.44 mL4.87 mL

*The above data is based on the productmolecular weight 410.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.