生物活性
Bexarotene (LGD1069)是一种高度选择性的类维生素A X受体（RXR）激动剂。
靶点信息
化学数据
| 目录号 | A11094 |
| M. Wt | 348.5 |
| Formula | C24H28O2 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
| CAS No. | 153559-49-0 |
| Synonyms | LGD 1069, SR 11247, Ro 26-4455, Targretin, LG 100069 |
| SMILES | CC1=CC2=C(C=C1C(=C)C3=CC=C(C=C3)C(=O)O)C(CCC2(C)C)(C)C |
溶解度
| In vitro | DMSO | 7 mg/mL (20.11 mM) |
| Water | Insoluble |
| Ethanol | Insoluble |
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
储备液配制
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
| 0.1 mM | 28.69 mL | 143.47 mL | 286.94 mL |
| 0.5 mM | 5.74 mL | 28.69 mL | 57.39 mL |
| 1 mM | 2.87 mL | 14.35 mL | 28.69 mL |
| 5 mM | 0.57 mL | 2.87 mL | 5.74 mL |
*The above data is based on the productmolecular weight 348.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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