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Lurasidone(SM13496)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Lurasidone(SM13496)图片
CAS NO:367514-87-2
包装与价格:
包装价格(元)
50mg电议
100mg电议
200mg电议

产品名称
SM13496, SM-13496, SM 13496
产品介绍

生物活性

Lurasidone (SM-13496)是dopamine D2和5-HT7的拮抗剂,IC50 值分别为 1.68 和 0.495 nM。Lurasidone (SM-13496) 也是 5-HT1A 受体的部分激动剂。

化学数据

目录号A11214
作用机制Inhibitor (抑制剂)
M. Wt492.7
FormulaC28H36N4O2S
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.367514-87-2
SynonymsSM13496, SM-13496, SM 13496
SMILESC1CC[C@H]([C@@H](C1)CN2CCN(CC2)C3=NSC4=CC=CC=C43)CN5C(=O)[C@H]6[C@@H]7CC[C@@H](C7)[C@H]6C5=O

溶解度

In vitroDMSO7 mg/mL (14.2 mM)
WaterInsoluble
EthanolInsoluble
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM20.3 mL101.48 mL202.96 mL
0.5 mM4.06 mL20.3 mL40.59 mL
1 mM2.03 mL10.15 mL20.3 mL
5 mM0.41 mL2.03 mL4.06 mL

*The above data is based on the productmolecular weight 492.7 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.