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Alvimopan(ADL 8-2698)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Alvimopan(ADL 8-2698)图片
CAS NO:156053-89-3
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议

产品名称
ADL 8-2698, Entereg, LY 246736
产品介绍

生物活性

Alvimopan (ADL 8-2698)表现为外周作用的opioid拮抗剂,Alvimopan竞争性结合胃肠道中的mu-opioid receptor。

化学数据

目录号A11292
作用机制Antagonist (拮抗剂)
M. Wt424.5
FormulaC25H32N2O4
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.156053-89-3
SynonymsADL 8-2698, Entereg, LY 246736
SMILESC[C@H]1CN(CC[C@@]1(C)C2=CC(=CC=C2)O)C[C@H](CC3=CC=CC=C3)C(=O)NCC(=O)O

溶解度

In vitroDMSO79 mg/mL (186.09 mM)
WaterInsoluble
EthanolInsoluble
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM23.56 mL117.79 mL235.57 mL
0.5 mM4.71 mL23.56 mL47.11 mL
1 mM2.36 mL11.78 mL23.56 mL
5 mM0.47 mL2.36 mL4.71 mL

*The above data is based on the productmolecular weight 424.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.