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L-689502
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
L-689502图片
CAS NO:138483-63-3
规格:98%
分子量:673.84
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议

产品介绍
L-689502是一个有效的HIV-1蛋白酶(HIV-lprotease)抑制剂,其IC50值为1nM。
CAS:138483-63-3
分子式:C39H51N3O7
分子量:673.84
纯度:98%
存储:Store at -20°C

Background:

L-689502 is a potent inhibitor of HIV-l protease with an IC50 of 1 nM.


Both L694746 and L-689502 inhibit HIV-l ptotease activity in a concentration-dependent manner. Pepstatin is much less potent than either compound exhibiting an IC50 of 2 μM. L694746 is as potent as L-689502 in inhibiting the HIV-l protease despite being structurally different from L-689502[1].



[1]. Lingham RB, et al. HIV-1 protease inhibitory activity of L-694,746, a novel metabolite of L-689,502. Biochem Biophys Res Commun. 1991 Dec 31;181(3):1456-61.