ML-10302 HCl is a potent 5-HT4 partial agonist (EC50 = 4 nM) that exhibits > 680-fold selectivity over 5-HT3 receptors (Kis are 1.07 and 730 nM respectively). References: Godínez-Chaparro B, López-Santillán FJ, Orduna P, Granados-Soto V. Secondary mechanical allodynia and hyperalgesia depend on descending facilitation mediated by spinal 5-HT4, 5-HT6 and 5-HT7 receptors. Neuroscience. 2012 Oct 11;222:379-91. doi: 10.1016/j.neuroscience.2012.07.008. PubMed PMID: 22796074.

纯度：≥98%

CAS：186826-17-5