CPUY074020 是一种有效的 G9a 抑制剂，IC50 值为 2.18 μM，具有抗增殖活性。
CAS：902279-44-1
分子式：C25H28N4O2
分子量：416.52
纯度：98%
存储：Store at -20°C

Background:

CPUY074020 is a potent G9a inhibitor with an IC50 of 2.18 μM, and possesses anti-proliferative activity [1]. IC50: 2.18 μM (G9a)[1]

[1]. Chen WL, et al. Discovery, design and synthesis of 6H-anthra[1,9-cd]isoxazol-6-one scaffold as G9a inhibitor through a combination of shape-based virtual screening and structure-based molecular. Bioorg Med Chem. 2016 Nov 15;24(22):6102-6108.