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(±)-Befunolol
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
(±)-Befunolol图片
CAS NO:39552-01-7
包装:1mg
规格:98%
市场价:2674元
分子量:291.34

产品介绍
(±)-Befunolol是一种β-肾上腺素能受体阻断剂。
CAS:39552-01-7
分子式:C16H21NO4
分子量:291.34
纯度:98%
存储:Store at -20°C

Background:

(±)-Befunolol is a β-adrenoceptor blocking agent.


A β-adrenoceptor blocking agent, Befunolol, is found to has intrinsic sympathomimetic activities in isolated right atria, trachea and taenia caecum of guinea pig (intrinsic activities are 0.22-0.28). The pD2-values of Befunolol estimated in the isolated organs are significantly different from its pA2-values against isoprenaline. Befunolol interacts with the beta-adrenoceptor where there may be two different sites: one site for agonistic action and the other for competitive antagonistic action. The intrinsic activity of Befunolol may be equal to its selectivity for both the sites[1].



[1]. Takayanagi I, et al. A beta-adrenoceptor blocking agent, befunolol as a partial agonist in isolated organs. Gen Pharmacol. 1985;16(3):265-7.