Epanolol(Visacor;ICI141292)是一种强效的β1-肾上腺素能受体激动剂。
CAS:86880-51-5
分子式:C20H23N3O4
分子量:369.41
纯度:98%
存储:Store at -20°C
Background:
Epanolol (Visacor; ICI141292) is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.
Epanolol is a novel anti-anginal agent which is a β1-adrenoceptor partial agonist exhibiting selective β1-adrenoceptor antagonist and selective β1-adrenoceptor agonist activity[1].
[1]. Hosie J, et al. Pharmacokinetics of epanolol after acute and chronic oral dosing in elderly patients with stable angina pectoris. Br J Clin Pharmacol. 1990 Mar;29(3):333-7.