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CYN 154806
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CYN 154806图片
CAS NO:183658-72-2
包装:1mg
规格:98%
市场价:3889元
分子量:1197.35

产品介绍
somatostatin sst2 receptor antagonist
CAS:183658-72-2
分子式:C56H68N12O14S2
分子量:1197.35
纯度:98%
存储:Store at -20°C

Background:

CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].


参考文献:
[1]. Bass RT, et al. Identification and characterization of novel somatostatin antagonists. Mol Pharmacol. 1996 Oct;50(4):709-15.
[2]. Feniuk W, et al. Selective somatostatin sst(2) receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology. 2000 Jun 8;39(8):1443-50.