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Salvinorin A Propionate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Salvinorin A Propionate图片
CAS NO:689295-71-4
规格:98%
分子量:446.5
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议

产品介绍
Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM.
CAS:689295-71-4
分子式:C24H30O8
分子量:446.5
纯度:98%
存储:Store at -20°C

Background:

Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM. It inhibits adenylate cyclase (EC50 = 4.7 nM) in HEK293 cells transfected with human KOR. It is selective for KORs over µ, δ, and ORL-1 opioid receptors and has no effect at serotonin, dopamine, muscarinic, or adrenergic receptors. In mice, salvinorin A propionate (13 µg, i.c.v.) reduces nociceptive responses in a radiant heat tail-flick assay, though not as potently as salvinorin A .