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Thrombin inhibitor 1
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Thrombin inhibitor 1图片
CAS NO:855998-46-8
规格:98%
分子量:497.32
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议

产品介绍
Thrombininhibitor1是一种有效的凝血酶抑制剂(Ki=0.66nM,2xaPTT=0.43μM)。
CAS:855998-46-8
分子式:C22H20Cl2F2N4O3
分子量:497.32
纯度:98%
存储:Store at -20°C

Background:

Thrombin inhibitor 1 is a potent thrombin inhibitor (Ki=0.66 nM, 2xaPTT=0.43 μM).


Thrombin inhibitor 1 (Compound 4) is binds in the active site of thrombin with Ki of 0.66 nM, 2xaPTT=0.43 uM). Thrombin inhibitor 1 (Compound 4) is evaluated for its thrombin inhibitory potency and its functional ability to double the activated partial thromboplastin time (2xaPTT) in human plasma with a 2xaPTT of 0.43 μM[1].



[1]. Nantermet PG, et al. P2 pyridine N-oxide thrombin inhibitors: a novel peptidomimetic scaffold. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2771-5.