Rilapladib是脂蛋白相关磷脂酶A2(Lp-PLA2)的一个选择性抑制剂，其IC50值为230pM。
CAS：412950-08-4
分子式：C40H38F5N3O3S
分子量：735.81
纯度：98%
存储：Store at -20°C

Background:

Rilapladib is a selective Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) inhibitor with an IC50 of 230 pM.

[1]. Shaddinger BC, et al. Platelet aggregation unchanged by lipoprotein-associated phospholipase A? inhibition: results from an in vitro study and two randomized phase I trials. PLoS One. 2014 Jan 27;9(1):e83094.