SOCE inhibitor 1是钙库调控的钙通道抑制剂,IC50为4.4 μM。
CAS:2169316-15-6
分子式:C25H22F3N5O4
分子量:513.47
纯度:98%
存储:Store at -20°C
Background:
SOCE inhibitor 1 is a store-operated calcium entry (SOCE) inhibitor with an IC50 of 4.4 μM.
IC50: 4.4 μM (SOCE)[1]
[1]. Riva B, et al. Pyrtriazoles, a Novel Class of Store-Operated Calcium Entry Modulators: Discovery, Biological Profiling, and in Vivo Proof-of-Concept Efficacy in Acute Pancreatitis. J Med Chem. 2018 Nov 8;61(21):9756-9783.