(1S,2S,3R)-DT-061是DT-061的对映异构体。DT-061是一种具有口服生物活性的、蛋白磷酸酶2A(PP2A)的激活剂，可用于治疗KRAS突变和MYC驱动的肿瘤。
CAS：1809427-20-0
分子式：C25H23F3N2O5S
分子量：520.52
纯度：98%
存储：Store at -20°C

Background:

(1S,2S,3R)-DT-061 is an enantiomer of DT-061. DT-061 is an orally bioavailable activator of protein phosphatase 2A (PP2A) and could be applied in the therapy of KRAS-mutant and MYC-driven tumorigenesis[1].

[1]. Kauko O, et al. PP2A inhibition is a druggable MEK inhibitor resistance mechanism in KRAS-mutant lung cancer cells. Sci Transl Med. 2018 Jul 18;10(450). pii: eaaq1093.