Drofenine盐酸盐是一种有效的竞争性胆碱酯酶抑制剂,ki值为3uM。
CAS:548-66-3
分子式:C20H32ClNO2
分子量:353.93
纯度:98%
存储:Store at -20°C
Background:
Drofenine hydrochloride is a potent competitive inhibitor of BChE, and the ki values of Drofenine is calculated to be 3 uM.IC50 value: 3 uM (ki)Target: BChEBenactyzine is widely used anticholinergic drugs, acts on smooth muscle to stop muscle spasms.
[1]. Bodur E, et al. Inhibition effects of benactyzine and drofenine on human serum butyrylcholinesterase. Arch Biochem Biophys. 2001 Feb 1;386(1):25-29.