c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate 是一种有效选择性的、短效肽的 V2 受体 (V2R) 激动剂,对 hV2R 和 rV2R 的 EC50 值分别为 0.07 和 0.02 nM。
CAS:1647120-04-4
分子式:C44H64ClN11O10S2
分子量:1006.63
纯度:98%
存储:Store at -20°C
Background:
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively[1].
EC50: 0.07 nM (hV2R), 0.02 nM (rV2R)[1]
[1]. Wi?niewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005.