GCN2-IN-1是一种有效的一般性调控阻遏蛋白激酶2(GCN2)抑制剂，在酶和细胞检测中IC50都<0.3μM。
CAS：1448693-69-3
分子式：C19H18N10O
分子量：402.41
纯度：98%
存储：Store at -20°C

Background:

GCN2-IN-1 is a potent general control nonderepressible 2 kinase (GCN2) inhibitor with IC50s of<0.3 μM in the enzyme and cell assay.

GCN2-IN-1 (Compound A-92) is a GCN2 inhibitor, which may be useful as a chemotherapeutic drug for the treatment of cancer[1].

[1]. Brazeau JF, et al. Triazolo[4,5-d]pyrimidine Derivatives as Inhibitors of GCN2. ACS Med Chem Lett. 2014 Feb 12;5(4):282-3.