A metabolite of dolutegravir
货号:ajcx25538
CAS:1485081-26-2
分子式:C13H15N3O5
分子量:293.3
溶解度:Methanol: slightly soluble
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Dolutegravir M1 is a metabolite of the HIV integrase inhibitor dolutegravir .1It is formed primarily by the cytochrome P450 (CYP) isoforms CYP1A1 and CYP1B1.
1.Zhu, J., Wang, P., Li, F., et al.CYP1A1 and 1B1-mediated metabolic pathways of dolutegravir, an HIV integrase inhibitorBiochem. Pharmacol.158174-184(2018)