STD1T 是一种脱泛素酶 USP2a 抑制剂,在 Ub-AMC 分析中, IC50 为 3.3 μM。
货号:ajcx33862
CAS:893075-58-6
分子式:C19H19N3O4S2
分子量:417.5
溶解度:DMSO : 62.5 mg/mL (149.70 mM; Need ultrasonic)
纯度:98%
存储:Store at -20°C
库存:
现货Background:
STD1T is a deubiquitinase USP2a inhibitor with an IC50 of 3.3 μM in Ub-AMC Assay[1].
STD1T inhibits USP2a enzymatic activity in a concentration dependent manner. STD1T shows selective inhibition of USP2a vs. USP7 at the concentrations of 10 µM and 2000 µM, respectively[1].
[1]. Marcin D Tomala, et al. Identification of small-molecule inhibitors of USP2a. Eur J Med Chem. 2018 Apr 25;150:261-267.