DS08210767 是一种高效的,具有生物口服可利用 PTHR1 拮抗剂,IC50 值为 90 nM。
货号:ajcx37350
CAS:2376334-75-5
分子式:C31H39N5O2
分子量:513.67
溶解度:N/A
纯度:98%
存储:Store at -20°C
库存:
现货Background:
DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM[1].
[1]. Arai Y, et al. Discovery of novel PTHR1 antagonists: Design, synthesis, and structure activity relationships. Bioorg Med Chem Lett. 2019 Sep 15;29(18):2613-2616.