Obafistat 是一种有效的醛酮还原酶 AKR1C3 抑制剂，对人 AKR1C3 的 IC50 值为 1.2 nM。
货号:ajcx35764
CAS:2160582-57-8
分子式:C15H16FN5O3S
分子量：365.38
溶解度:DMSO : 62.5 mg/mL (171.05 mM; ultrasonic and warming and heat to 60°C)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Obafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC50 of 1.2 nM for human AKR1C3 (patent WO2017202817A1, example 4)[1].

[1]. Marcus Koppitz, et al. [8-(phenylsulfonyl)-3,8-diazabicyclo[3.2.1]oct-3-yl] (1h-1,2,3-triazol-4-yl)methanones. WO2017202817A1.