ElacestrantSenantiomerdihydrochloride(RAD1901Senantiomerdihydrochloride)是Elacestrant的低活性对映体。Elacestrant(RAD1901)dihydrochloride是有选择性和口服活性的雌激素受体(ER)的降解剂,对ERα和ERβ的IC50值分别为48和870nM。
货号:ajcx30576
CAS:2309762-30-7
分子式:C30H40Cl2N2O2
分子量:531.56
溶解度:N/A
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Elacestrant S enantiomer dihydrochloride (RAD1901 S enantiomer dihydrochloride) is an low activity enantiomer of elacestrant dihydrochloride. Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.