Enzalutamide D3 是一种氘标记的 Enzalutamide (MDV3100)。Enzalutamide 是一种雄激素受体 (AR) 拮抗剂,在 LNCaP 前列腺细胞中 IC50 为 36 nM。
货号:ajcx38426
CAS:1443331-82-5
分子式:C21H13D3F4N4O2S
分子量:467.45
溶解度:N/A
纯度:98%
存储:Store at -20°C
库存:
现货Background:
Enzalutamide D3 is a deuterium labeled Enzalutamide (MDV3100). Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells[1].
[1]. Tran C, et al. Development of a second-generation antiandrogen for treatment of advanced prostate cancer. Science. 2009 May 8;324(5928):787-90.