An inhibitor of ASK1
货号:ajcx22030
CAS:2411382-24-4
分子式:C19H19N9O2
分子量:405.4
溶解度:Chloroform: 10 mg/ml
纯度:98%
存储:Store at -20°C
库存:
现货Background:
CAY10756 is a brain-penetrant inhibitor of apoptosis signal-regulating kinase 1 (ASK1; IC50= 21 nM).1It inhibits autophosphorylation of ASK1 in HEK293T cells (IC50= 138 nM).
1.Xin, Z., Himmelbauer, K., Jones, J.H., et al.Discovery of CNS-penetrant apoptosis signal-regulating kinase 1 (ASK1) inhibitorsACS Med. Chem. Lett.11(4)485-490(2020)