Takeda103A 是一种有效的 GRK2 抑制剂。G 蛋白偶联受体 (GPCR) 是许多生理过程的核心。Takeda103A 具有研究心力衰竭的潜力。
货号:ajcx39628
CAS:865609-72-9
分子式:C24H23F2N7O
分子量：463.48
溶解度:N/A
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Takeda103A is a potent inhibitor of GRK2. G protein-coupled receptors (GPCRs) are central to many physiological processes. Takeda103A has the potential for the research of heart failure[1].

[1]. Waldschmidt HV, et al. Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors. J Med Chem. 2016;59(8):3793-3807.