KHK-IN-2是有效,选择性的果糖激酶 (KHK)抑制剂,IC50为 0.45 μM。
货号:ajcx39488
CAS:2135304-43-5
分子式:C16H19F3N4O3
分子量:372.34
溶解度:DMSO : 250 mg/mL (671.43 mM; Need ultrasonic)
纯度:98%
存储:Store at -20°C
库存:
现货Background:
KHK-IN-2 is a potent and selective ketohexokinase (KHK) inhibitor with an IC50 of 0.45 μM.
[1]. Huard K, et al. Discovery of Fragment-Derived Small Molecules for in Vivo Inhibition of Ketohexokinase (KHK). J Med Chem. 2017 Sep 28;60(18):7835-7849.